Reference

Drug formulary

Every agent in the chapter in one place. Filter by drug class or by treatment horizon — acute/symptomatic versus maintenance/targeted — to compare indication, dose, mechanism, cautions and the strength of the evidence.

Drug formulary

27 of 27 agents
  • MeclizineAntihistamineSymptomatic only
    For
    Acute peripheral vertigo, motion sickness
    Dose
    25–50 mg PO 2–3×/day
    Mechanism
    H1 antagonist with weak anticholinergic action; dampens vestibular-nucleus signalling
    Cautions
    Sedation (less than others), dry mouth; safer choice in pregnancy (FDA category B)
  • DimenhydrinateAntihistamineSymptomatic only
    For
    Acute vertigo with nausea, motion sickness
    Dose
    50–100 mg PO every 4–6 h
    Mechanism
    Diphenhydramine + chlorotheophylline salt; H1/anticholinergic, fast onset
    Cautions
    Marked sedation; limit in older adults and tasks needing alertness
  • PromethazineAntihistamineSymptomatic only
    For
    Acute vertigo with intractable nausea/vomiting (ED)
    Dose
    12.5–25 mg PO/IM
    Mechanism
    Phenothiazine H1 antagonist with potent antiemetic and sedative effect
    Cautions
    Deep sedation, extrapyramidal symptoms
  • DiphenhydramineAntihistamineSymptomatic only
    For
    Acute vertigo / nausea (selected)
    Dose
    25–50 mg PO/IM
    Mechanism
    First-generation ethanolamine H1 antagonist
    Cautions
    High anticholinergic load and sedation; avoid in older adults, urinary retention, cognitive impairment
  • Scopolamine (hyoscine)AnticholinergicModerate
    For
    Prophylaxis of motion sickness
    Dose
    1.5 mg transdermal patch / 72 h behind the ear
    Mechanism
    Blocks M1 muscarinic receptors in vestibular nuclei, reticular formation and CTZ
    Cautions
    Confusion, delirium, dry mouth, blurred vision, urinary retention; avoid in elderly, glaucoma, BPH
  • DiazepamBenzodiazepineSymptomatic only
    For
    Severe acute vertigo (e.g. neuritis, Ménière's attack)
    Dose
    2–10 mg PO twice daily (short course)
    Mechanism
    GABA-A potentiation → suppresses vestibular-nucleus firing; rapid onset, long half-life
    Cautions
    Sedation, falls, dependence; delays central compensation — limit to 3–5 days
  • LorazepamBenzodiazepineSymptomatic only
    For
    Acute vertigo, intermediate duration
    Dose
    0.5–2 mg PO twice daily (short course)
    Mechanism
    GABA-A potentiation; shorter half-life than diazepam
    Cautions
    Sedation, dependence; limit duration, avoid during vestibular rehabilitation
  • ClonazepamBenzodiazepineLimited
    For
    Vestibular hypersensitivity, vestibular migraine, functional dizziness
    Dose
    0.25–0.5 mg PO twice daily
    Mechanism
    GABA-A potentiation with anxiolytic effect; reduces visual dependence
    Cautions
    Sedation, tolerance, dependence; not for chronic maintenance
  • ProchlorperazineDopamine antagonistSymptomatic only
    For
    Vertigo-induced nausea and vomiting
    Dose
    5–10 mg PO/IM three times daily
    Mechanism
    Blocks D2 receptors in the chemoreceptor trigger zone
    Cautions
    Extrapyramidal symptoms (dystonia, parkinsonism); short-term use only
  • MetoclopramideDopamine antagonistSymptomatic only
    For
    Vertigo-associated nausea/vomiting
    Dose
    10 mg PO/IV three times daily
    Mechanism
    Central + peripheral D2 antagonist; prokinetic antiemetic
    Cautions
    Extrapyramidal symptoms, especially in children and with prolonged use
  • BetahistineHistamine analogueModerate
    For
    Ménière's disease — prophylaxis of attacks
    Dose
    16–48 mg/day in divided doses
    Mechanism
    Weak H1 agonist + potent H3 antagonist; improves inner-ear microcirculation and endolymph resorption
    Cautions
    Generally well tolerated; caution in active peptic ulcer, asthma. Audiological benefit inconsistent
  • Hydrochlorothiazide + triamtereneDiureticLimited
    For
    Ménière's disease — adjunct with low-sodium diet
    Dose
    One tablet daily (with diet < 1.5 g sodium/day)
    Mechanism
    Reduces body fluid volume → theoretically lowers endolymphatic pressure
    Cautions
    Electrolyte imbalance, dehydration, hypotension; monitor renal function. Evidence largely observational
  • AcetazolamideDiureticLimited
    For
    Ménière's disease (selected); some episodic ataxias
    Dose
    250–500 mg/day
    Mechanism
    Carbonic anhydrase inhibitor; mild diuresis and metabolic acidosis
    Cautions
    Paraesthesiae, electrolyte disturbance; limited Ménière's evidence
  • Prednisone / methylprednisolone (oral)CorticosteroidModerate
    For
    Vestibular neuritis — accelerate recovery
    Dose
    Prednisone 60 mg/day, tapered over 10–14 days; start < 72 h
    Mechanism
    Anti-inflammatory; reduces vestibular-nerve oedema and improves caloric recovery
    Cautions
    Hyperglycaemia, GI irritation, immunosuppression; functional benefit debated
  • IV methylprednisoloneCorticosteroidEstablished
    For
    MS relapse causing central vertigo
    Dose
    1 g/day IV for 3–5 days (± oral taper)
    Mechanism
    High-dose anti-inflammatory; stabilises blood–brain barrier, shortens relapse
    Cautions
    Hyperglycaemia, mood change, infection risk; does not alter long-term MS course
  • Intratympanic steroidIntratympanicModerate
    For
    Refractory Ménière's disease (hearing-sparing)
    Dose
    Dexamethasone / methylprednisolone via round window
    Mechanism
    Local anti-inflammatory; stabilises membrane permeability with minimal systemic effect
    Cautions
    Procedural; efficacy varies between individuals
  • Intratympanic gentamicinIntratympanicModerate
    For
    Refractory disabling Ménière's vertigo
    Dose
    Titrated aminoglycoside via round window
    Mechanism
    Vestibulotoxic chemical ablation of vestibular hair cells (> 85% vertigo control)
    Cautions
    Risk of cochleotoxicity / hearing loss and persistent imbalance; specialist-administered
  • SumatriptanMigraine — acuteLimited
    For
    Acute vestibular migraine attack
    Dose
    Per migraine protocol, taken early in the episode
    Mechanism
    5-HT1B/1D agonist; reduces neurogenic inflammation and trigeminovascular signalling
    Cautions
    Cardiovascular contraindications; efficacy in VM more variable than in migraine with aura
  • PropranololMigraine — prophylaxisModerate
    For
    Vestibular migraine prophylaxis
    Dose
    40–160 mg/day
    Mechanism
    β-blocker; modulates adrenergic tone and cerebrovascular reactivity
    Cautions
    Bradycardia, fatigue, bronchospasm; avoid in asthma
  • FlunarizineMigraine — prophylaxisModerate
    For
    Vestibular migraine prophylaxis (RCT-supported)
    Dose
    10 mg/day
    Mechanism
    Calcium-channel blocker; stabilises vestibular neurons and reduces excitability
    Cautions
    Weight gain, sedation, depression, parkinsonism with long use
  • AmitriptylineMigraine — prophylaxisLimited
    For
    VM with coexisting tension headache, insomnia or anxiety
    Dose
    10–50 mg at bedtime
    Mechanism
    Tricyclic; inhibits serotonin/noradrenaline reuptake, modulating pain pathways
    Cautions
    Anticholinergic effects, sedation, QT prolongation
  • TopiramateMigraine — prophylaxisModerate
    For
    Vestibular migraine prophylaxis, refractory cases
    Dose
    25–100 mg/day
    Mechanism
    Modulates Na/Ca channels and enhances GABAergic inhibition
    Cautions
    Paraesthesiae, cognitive slowing, weight loss, teratogenicity
  • SertralineSSRI / SNRIModerate
    For
    PPPD — first-line
    Dose
    50–200 mg/day (start low, titrate)
    Mechanism
    Enhances serotonergic transmission in vestibular nuclei and parieto-insular cortex; reduces visual dependence
    Cautions
    Nausea, headache, sexual dysfunction; benefit takes 4–6 weeks
  • ParoxetineSSRI / SNRIModerate
    For
    PPPD — RCT-supported (60–70% improvement)
    Dose
    10–40 mg/day
    Mechanism
    SSRI; desensitises abnormal vestibulo-visual responses and motion-triggered anxiety
    Cautions
    Anticholinergic and discontinuation effects; titrate and taper
  • VenlafaxineSSRI / SNRIModerate
    For
    PPPD — most-used SNRI
    Dose
    75–150 mg/day
    Mechanism
    SNRI; serotonergic/noradrenergic modulation of central vestibular processing
    Cautions
    Hypertension at higher doses, nausea, discontinuation syndrome
  • GabapentinOther / emergingLimited
    For
    Symptomatic nystagmus (e.g. in MS), some central vertigo
    Dose
    Titrated to effect
    Mechanism
    Modulates voltage-gated calcium channels; suppresses pathological nystagmus
    Cautions
    Sedation, dizziness, ataxia
  • MemantineOther / emergingLimited
    For
    Pendular nystagmus; investigational for central imbalance
    Dose
    Titrated to effect
    Mechanism
    NMDA-receptor antagonist; modulates central vestibular plasticity
    Cautions
    Dizziness, headache; role in vertigo not yet established
Doses are illustrative teaching figures, not prescribing instructions — verify every drug, dose and contraindication against the current formulary and the individual patient. Evidence grades are a pragmatic teaching summary: Established › Moderate › Limited › Symptomatic only.

For learning, not prescribing.Doses are illustrative teaching figures. Always verify the drug, dose, interactions and contraindications against the current formulary and the individual patient, and remember the chapter’s governing rule — symptomatic suppressants are for the first 3–5 days only.